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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T13105 | TD-428 | Epigenetic Reader Domain | |
TD-428 is a highly specific degrader of BRD4(DC50 of 0.32 nM). TD-428 is a BET PROTAC, which comprises TD-106 (a CRBN ligand) linked to JQ1 (a BET inhibitor). TD-428 efficiently induce BET protein degradation. |